SCHEMBL12176643

SCHEMBL12176643

BCCc1cccc(-c2nnc(-c3ccc(CC(C)C)c(N)c3)s2)c1CC

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 18/20 0.46
S1PR3 Q99500 1/20 0.37
CYP2C9 P11712 4/20 0.34
NOTUM Q6P988 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12176514 0.92 S1PR1 (0.43) S1PR1S1PR3CYP2C9NOTUM
SCHEMBL12102825 0.85 S1PR1 (0.58) S1PR1S1PR3CYP2C9
SCHEMBL12176280 0.83 S1PR1 (0.58) S1PR1S1PR3CYP2C9
SCHEMBL12102741 0.77 S1PR1 (0.56) S1PR1S1PR3CYP2C9
SCHEMBL12102768 0.77 S1PR1 (0.59) S1PR1S1PR3CYP2C9
SCHEMBL13974005 0.76 S1PR1 (0.59) S1PR1S1PR3CYP2C9
SCHEMBL12175443 0.75 S1PR1 (0.54) S1PR1S1PR3
SCHEMBL12102428 0.71 S1PR1 (0.42) S1PR1S1PR3CYP2C9
SCHEMBL1293239 0.71 S1PR1 (0.55) S1PR1S1PR3CYP2C9
SCHEMBL12176644 0.71 S1PR1 (0.58) S1PR1S1PR3CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011134280-A1 COMPOUNDS AS AGONISTS OF S1P1 RECEPTORS GLAXO GROUP LIMITED (GB) 2011-11-03 WO disclosed