SCHEMBL13985463

SCHEMBL13985463

CC(C)(C)OC(=O)NCc1ccc(-c2nc3c(N4CCN(Cc5cncc(F)c5)CC4)c(Br)cnc3[nH]2)cc1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AURKA O14965 15/20 0.42
GNRHR P30968 2/20 0.39
IGF1R P08069 1/20 0.39
ROCK2 O75116 1/20 0.38
KIT P10721 1/20 0.38
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13985729 0.89 TBK1 (0.44) AURKAGNRHR
SCHEMBL211207 0.89 AURKA (0.53) AURKAGNRHRIGF1RCYP1A2CYP2D6
SCHEMBL13985706 0.87 AURKA (0.44) AURKAGNRHRKCNH2
SCHEMBL13985592 0.86 TBK1 (0.42) AURKAGNRHRIGF1RROCK2
SCHEMBL13985737 0.84 AURKA (0.55) AURKAKCNH2
SCHEMBL210188 0.83 AURKA (0.48) AURKAGNRHRIGF1RROCK2KIT
SCHEMBL13985464 0.83 AURKA (0.50) AURKAGNRHRCYP1A2CYP2D6CYP2C9
SCHEMBL4754714 0.82 AURKA (0.52) AURKACYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL13985645 0.81 AURKA (0.51) AURKACYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL13985468 0.79 AURKA (0.41) AURKAIGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001021-A1 IMIDAZOPYRIDINE DERIVATIVES USEFUL AS ENZYME INHIBITORS FOR THE TREATMENT OF CELL PROLIFERATIVE AND AUTOIMMUNE DISEASES CHROMA THERAPEUTICS LTD. (GB) 2008-12-31 WO disclosed