SCHEMBL13985474

SCHEMBL13985474

NCc1ccc(-c2nc3c(N4CCN(Cc5cccnc5)CC4)c(Cl)cnc3[nH]2)cc1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AURKA O14965 13/20 0.52
DRD2 P14416 3/20 0.47
DRD4 P21917 3/20 0.47
DRD3 P35462 3/20 0.47
CYP2D6 P10635 2/20 0.45
CYP2C9 P11712 2/20 0.45
CYP2C19 P33261 2/20 0.45
KCNH2 Q12809 2/20 0.45
CYP1A2 P05177 1/20 0.45
GNRHR P30968 1/20 0.42
KDR P35968 1/20 0.41
AURKB Q96GD4 1/20 0.41
CASP1 P29466 1/20 0.40
CASP4 P49662 1/20 0.40
CASP5 P51878 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL210671 0.90 AURKA (0.64) AURKADRD2DRD4DRD3CYP2D6
SCHEMBL14495854 0.89 AURKA (0.50) AURKADRD2DRD4DRD3CYP2D6
SCHEMBL210273 0.89 AURKA (0.61) AURKADRD2DRD4DRD3CYP2D6
SCHEMBL210907 0.88 AURKA (0.54) AURKADRD2DRD4DRD3CYP2D6
SCHEMBL211945 0.87 AURKA (0.50) AURKADRD2DRD4DRD3CYP2D6
SCHEMBL4756520 0.87 AURKA (0.48) AURKADRD2DRD4DRD3CYP2D6
SCHEMBL4757490 0.86 AURKA (0.50) AURKADRD2DRD4DRD3KCNH2
SCHEMBL13985732 0.84 AURKA (0.48) AURKACYP2D6CYP2C9CYP2C19KCNH2
SCHEMBL211129 0.84 AURKA (0.48) AURKADRD2DRD4DRD3CYP2D6
SCHEMBL13985593 0.83 AURKA (0.45) AURKADRD2DRD4DRD3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001021-A1 IMIDAZOPYRIDINE DERIVATIVES USEFUL AS ENZYME INHIBITORS FOR THE TREATMENT OF CELL PROLIFERATIVE AND AUTOIMMUNE DISEASES CHROMA THERAPEUTICS LTD. (GB) 2008-12-31 WO disclosed