SCHEMBL13987828

SCHEMBL13987828

CCOC(=O)c1cc(-c2ccnc(Cl)c2)c[nH]1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNC P24863 4/20 0.64
CDK8 P49336 4/20 0.64
CDK5 Q00535 1/20 0.46
CDK5R1 Q15078 1/20 0.46
MMP2 P08253 2/20 0.44
MMP13 P45452 2/20 0.44
MMP14 P50281 2/20 0.44
ALPL P05186 1/20 0.44
GABRP O00591 1/20 0.42
GABRD O14764 1/20 0.42
GABRA1 P14867 1/20 0.42
GABRB1 P18505 1/20 0.42
GABRG2 P18507 1/20 0.42
GABRB3 P28472 1/20 0.42
GABRA5 P31644 1/20 0.42
GABRA3 P34903 1/20 0.42
GABRA2 P47869 1/20 0.42
GABRB2 P47870 1/20 0.42
GABRA4 P48169 1/20 0.42
GABRE P78334 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16116380 0.85 CCNC (0.68) CCNCCDK8ALDH1A1LMNAGAA
SCHEMBL4717248 0.81 ALPL (0.69) CDK5CDK5R1ALPLNPC1ALDH1A1
SCHEMBL1126787 0.80 NOTUM (0.60) ALPLGABRPGABRDGABRA1GABRB1
SCHEMBL13987890 0.79 CCNC (0.76) CCNCCDK8ALPL
SCHEMBL4890571 0.79 SYK (0.53) NPC1HPGDRAB9ASMN1; SMN2
SCHEMBL1990531 0.79 JAK2 (0.53) ALPLGABRPGABRDGABRA1GABRB1
Lithium SCHEMBL16116438 0.78 CCNC (0.74) CCNCCDK8ALPL
SCHEMBL16116435 0.78 CCNC (0.74) CCNCCDK8ALPL
SCHEMBL16115998 0.78 CCNC (1.00) CCNCCDK8ALDH1A1RAB9AKMT2A
Lithium Ion SCHEMBL16116436 0.77 CCNC (0.72) CCNCCDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7462612-B2 Pyridine inhibitors of ERK2 and uses thereof VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-12-09 US disclosed
US-7462612-B2 Pyridine inhibitors of ERK2 and uses thereof VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-12-09 US disclosed