SCHEMBL13999992

SCHEMBL13999992

CC(C)C1ON=C(c2c(Cl)cccc2Cl)C1COc1ccc(-c2ccc3c(C(=O)O)c[nH]c3c2)cc1

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 5/20 0.59
PRKAB2 O43741 15/20 0.47
PRKAG1 P54619 15/20 0.47
PRKAA2 P54646 15/20 0.47
PRKAA1 Q13131 15/20 0.47
PRKAG3 Q9UGI9 15/20 0.47
PRKAG2 Q9UGJ0 15/20 0.47
PRKAB1 Q9Y478 15/20 0.47
NR1I2 O75469 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13999486 0.86 PRKAG1 (0.47) NR1H4PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL14215772 0.85 NR1H4 (0.59) NR1H4NR1I2CYP1A2CYP3A4CYP2C9
SCHEMBL13999489 0.85 NR1H4 (0.60) NR1H4NR1I2CYP1A2CYP3A4CYP2C9
SCHEMBL13999491 0.84 NR1H4 (0.42) NR1H4NR1I2CYP1A2CYP3A4CYP2C9
SCHEMBL14215895 0.84 NR1H4 (0.46) NR1H4NR1I2CYP1A2CYP3A4CYP2C9
SCHEMBL13999479 0.84 NR1H4 (0.59) NR1H4NR1I2CYP1A2CYP3A4CYP2C9
SCHEMBL14215811 0.82 NR1H4 (0.59) NR1H4NR1I2CYP1A2CYP3A4CYP2C9
SCHEMBL13999592 0.82 NR1H4 (0.59) NR1H4NR1I2CYP1A2CYP3A4CYP2C9
SCHEMBL14215784 0.81 NR1H4 (0.46) NR1H4NR1I2CYP1A2CYP3A4CYP2C9
SCHEMBL13999579 0.81 NR1H4 (0.46) NR1H4NR1I2CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008157270-A1 FARNESOID X RECEPTOR AGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-24 WO disclosed