SCHEMBL14000815

SCHEMBL14000815

O=C(NC1CCNCC1)c1ccc(-n2cc3ccccc3n2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GCG P01275 2/20 0.52
KHK P50053 3/20 0.50
RAB9A P51151 2/20 0.45
MAPT P10636 1/20 0.45
HDAC4 P56524 2/20 0.44
HDAC6 Q9UBN7 2/20 0.44
PARP1 P09874 1/20 0.43
ACSS2 Q9NR19 1/20 0.43
SMYD3 Q9H7B4 2/20 0.43
GCGR P47871 1/20 0.43
HTR4 Q13639 2/20 0.43
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
FLT3 P36888 1/20 0.41
ACP1 P24666 1/20 0.41
HPGDS O60760 1/20 0.41
PTK2 Q05397 1/20 0.41
HDAC3 O15379 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14000452 0.93 GCG (0.50) GCGKHKRAB9AMAPTHDAC4
Tert-Butyl Formate SCHEMBL27808400 0.89 GCG (0.46) GCGKHKRAB9AMAPTHDAC4
SCHEMBL3723766 0.79 HDAC4 (0.54) GCGHDAC4HDAC6PARP1KMT2A
SCHEMBL3668247 0.78 HRH3 (0.44) PARP1PTK2
SCHEMBL3730320 0.75 HDAC4 (0.55) GCGHDAC4HDAC6PARP1
SCHEMBL4946424 0.75 HDAC4 (0.55) GCGHDAC4HDAC6PARP1
SCHEMBL27786338 0.74 GCG (0.44) GCGPARP1GCGRNPC1HPGDS
SCHEMBL594567 0.74 NPC1 (0.62) KHKRAB9AHDAC4HDAC6SMYD3
SCHEMBL3667714 0.74 SLC6A4 (0.45)
SCHEMBL3666843 0.74 SLC6A4 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008147945-A1 AZACYCLYLBENZAMIDE DERIVATIVES AS HISTAMINE-3 ANTAGONISTS WYETH (US) 2008-12-04 WO disclosed