SCHEMBL14010989

SCHEMBL14010989

C/C=C/c1ccc(C(C)(C)O)cc1F

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 2/20 0.37
CYP1B1 Q16678 2/20 0.37
CYP1A2 P05177 1/20 0.36
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
NFE2L2 Q16236 4/20 0.34
MIF P14174 1/20 0.34
PDE2A O00408 4/20 0.33
TNKS O95271 3/20 0.33
PARP1 P09874 3/20 0.33
TNKS2 Q9H2K2 3/20 0.33
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33
PDE10A Q9Y233 2/20 0.32
F2RL1 P55085 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12732541 1.00 CYP1A1 (0.37) CYP1A1CYP1B1CYP1A2PTGS1PTGS2
SCHEMBL13841271 0.81 CYP1A1 (0.45) CYP1A1CYP1B1NFE2L2PDE2A
SCHEMBL1673838 0.81 CYP1A1 (0.40) CYP1A1CYP1B1CYP1A2PTGS1PTGS2
SCHEMBL1673839 0.81 CYP1A1 (0.40) CYP1A1CYP1B1CYP1A2PTGS1PTGS2
SCHEMBL1246657 0.80 TNKS (0.37) CYP1A1CYP1B1PDE2ATNKSPARP1
SCHEMBL12663410 0.76
SCHEMBL6967423 0.74 KCNN4 (0.43) PDE2ATNKSPARP1TNKS2
SCHEMBL12732543 0.73 GPR183 (0.39) CYP1A1CYP1B1CYP1A2PTGS1PTGS2
SCHEMBL7651798 0.72 NFE2L2 (0.61) CYP1A1CYP1B1PTGS1PTGS2NFE2L2
SCHEMBL13891146 0.72 NFE2L2 (0.61) CYP1A1CYP1B1PTGS1PTGS2NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008156726-A1 INHIBITORS OF JANUS KINASES MERCK & CO., INC. (US) 2008-12-24 WO disclosed