SCHEMBL14014336

SCHEMBL14014336

Cn1c(Nc2cc(F)c(I)cc2F)c(C(N)=O)c(=O)n(C)c1=O

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.37
MAP2K1 Q02750 18/20 0.37
MAP2K2 P36507 6/20 0.37
MAPT P10636 1/20 0.36
MAP2K5 Q13163 1/20 0.35
EIF2AK1 Q9BQI3 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL217405 0.84 MAP2K1 (0.54) MAP2K1MAP2K2MAP2K5EIF2AK1
SCHEMBL14647529 0.81 MAP2K1 (0.54) HTTMAP2K1MAP2K2MAPTMAP2K5
SCHEMBL220490 0.80 MAP2K1 (0.55) HTTMAP2K1MAP2K2
SCHEMBL221014 0.79 MAP2K1 (0.58) MAP2K1MAP2K2MAP2K5
SCHEMBL221013 0.79 MAP2K1 (0.58) MAP2K1MAP2K2MAP2K5
SCHEMBL219481 0.78 IDO1 (0.41) HTTMAP2K1MAP2K2MAPTMAP2K5
SCHEMBL3010504 0.73 MAP2K1 (0.58) MAP2K1MAP2K2MAP2K5EIF2AK1
SCHEMBL218724 0.73 MAP2K1 (0.58) MAP2K1MAP2K2MAP2K5EIF2AK1
SCHEMBL27765754 0.73 MAP2K1 (0.37) MAP2K1MAP2K2MAP2K5EIF2AK1
SCHEMBL218385 0.73 MAP2K1 (0.52) MAP2K1MAP2K2MAP2K5EIF2AK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008140553-A2 MAPK/ERK KINASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-11-20 WO disclosed