SCHEMBL14016409

SCHEMBL14016409

c1ccc(CN2CC34CNCC3(C2)CN(Cc2ccccc2)C4)cc1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.55
GAA P10253 1/20 0.53
TSHR P16473 3/20 0.50
CYP2D6 P10635 2/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
ALDH1A1 P00352 2/20 0.50
CYP3A4 P08684 2/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
HIF1A Q16665 1/20 0.50
TDP1 Q9NUW8 1/20 0.47
HSD17B10 Q99714 1/20 0.46
MC4R P32245 1/20 0.46
KDM4E B2RXH2 1/20 0.44
MAPT P10636 1/20 0.44
HTT P42858 1/20 0.44
DRD4 P21917 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15985246 0.86 CYP2D6 (0.60) SIGMAR1GAATSHRCYP2D6MEN1
SCHEMBL29598556 0.86 GAA (0.61) SIGMAR1GAATSHRCYP2D6MEN1
Hydrochloric Acid SCHEMBL31645775 0.85 CYP2D6 (0.59) SIGMAR1GAATSHRCYP2D6MEN1
Oxalic Acid SCHEMBL20798190 0.83 CYP2D6 (0.54) SIGMAR1GAATSHRCYP2D6MEN1
SCHEMBL14016365 0.79 GAA (0.46) SIGMAR1GAATSHRCYP2D6MEN1
SCHEMBL27798357 0.79 SIGMAR1 (0.62) SIGMAR1GAATSHRCYP2D6MEN1
SCHEMBL11707747 0.78 GAA (0.61) SIGMAR1GAATSHRCYP2D6MEN1
SCHEMBL4588336 0.78 TSHR (0.40) SIGMAR1GAATSHRCYP2D6MEN1
SCHEMBL4292159 0.77 CYP2D6 (0.76) SIGMAR1TSHRCYP2D6MEN1KMT2A
SCHEMBL1426377 0.77 CYP2D6 (0.67) SIGMAR1GAATSHRCYP2D6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7435831-B2 Bicyclic and bridged nitrogen heterocycles CHEMOCENTRYX, INC. (US) 2008-10-14 US disclosed
WO-2007027734-A2 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX, INC. (US) 2007-03-08 WO disclosed