SCHEMBL14017159

SCHEMBL14017159

CN(C)C1CCN(C(=O)[C@@H](Cc2cc(C(F)(F)F)c(N)c(C(F)(F)F)c2)NC(=O)N2CCC(N3Cc4ccccc4NC3=O)CC2)CC1

nearest known ligand 0.60

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CALCA P06881 1/20 0.60
CALCRL Q16602 18/20 0.57
CYP3A4 P08684 16/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14016933 0.96 CALCA (0.65) CALCACALCRLCYP3A4
SCHEMBL14017063 0.95 CALCRL (0.58) CALCACALCRLCYP3A4
SCHEMBL13331687 0.94 CALCRL (0.58) CALCACALCRLCYP3A4
SCHEMBL14016744 0.91 CALCRL (0.70) CALCRLCYP3A4
SCHEMBL14017026 0.90 CALCA (0.61) CALCACALCRLCYP3A4
SCHEMBL3961490 0.90 CALCA (0.70) CALCACALCRLCYP3A4
SCHEMBL13713222 0.90 CALCA (0.57) CALCACALCRLCYP3A4
SCHEMBL13331861 0.90 CALCA (0.57) CALCACALCRLCYP3A4
SCHEMBL13713157 0.90 CALCRL (0.56) CALCACALCRLCYP3A4
SCHEMBL3309830 0.89 CALCRL (0.65) CALCACALCRLCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7439237-B2 Selected CGRP-antagonists, process for preparing them and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-10-21 US disclosed