SCHEMBL14018552

SCHEMBL14018552

COC(=O)c1ccc(/C=C/c2cc3c(cc2/C=C/S(N)(=O)=O)C(C)(C)CCC3(C)C)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 6/20 0.52
RARG P13631 6/20 0.52
RARA P10276 5/20 0.52
PTPN1 P18031 1/20 0.47
VDR P11473 4/20 0.45
CYP3A4 P08684 3/20 0.45
STS P08842 1/20 0.44
CYP26A1 O43174 3/20 0.42
NPC1 O15118 2/20 0.41
LMNA P02545 2/20 0.41
MAPT P10636 2/20 0.41
MEN1 O00255 1/20 0.41
S1PR4 O95977 1/20 0.41
ALDH1A1 P00352 1/20 0.41
POLB P06746 1/20 0.41
ALPG P10696 1/20 0.41
THRB P10828 1/20 0.41
PKM P14618 1/20 0.41
S1PR1 P21453 1/20 0.41
NTSR1 P30989 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14017812 0.90 RARB (0.53) RARBRARGRARAPTPN1VDR
SCHEMBL14159883 0.87 RARB (0.68) RARBRARGRARACYP3A4CYP26A1
SCHEMBL2594345 0.82 RARB (0.75) RARBRARGRARAPTPN1VDR
SCHEMBL4666958 0.82 RARB (0.75) RARBRARGRARAPTPN1VDR
SCHEMBL14018613 0.82 RARB (0.60) RARBRARGRARACYP3A4CYP26A1
SCHEMBL10842924 0.81 RARB (0.55) RARBRARGRARAPTPN1VDR
SCHEMBL10842927 0.81 RARB (0.55) RARBRARGRARAPTPN1VDR
SCHEMBL14159774 0.80 RARB (0.52) RARBRARGRARAPTPN1VDR
SCHEMBL1615332 0.80 RARB (0.72) RARBRARGRARAPTPN1VDR
SCHEMBL1615774 0.80 RARB (0.72) RARBRARGRARAPTPN1VDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1324970-B1 RETINOIDS FOR THE TREATMENT OF EMPHYSEMA HOFFMANN LA ROCHE (CH) 2008-11-05 EP disclosed
EP-1935869-A1 Retinoids for the treatment of emphysema F. HOFFMANN-LA ROCHE AG (CH) 2008-06-25 EP disclosed