SCHEMBL1402086

SCHEMBL1402086

CCCN(C(=O)C(F)(F)F)[C@H]1C[C@@H](n2cnc3c(NCCC(C)(C)C)nc(N4CC[C@@H](NC(=O)NC5CCNC5)C4)nc32)[C@H](O)[C@H]1O

nearest known ligand 0.31

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.31
HRH4 Q9H3N8 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
CNR2 P34972 1/20 0.31
CDK1 P06493 1/20 0.30
CDK5 Q00535 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2091171 1.00 ADORA2A (0.31) ADORA2AHRH4HRH3CNR2CDK1
SCHEMBL1402056 0.91 ADORA2A (0.38) ADORA2ACDK1CDK5
SCHEMBL1402089 0.91 ADORA2A (0.36) ADORA2A
SCHEMBL1402138 0.90 CDK1 (0.33) ADORA2AHRH4HRH3CNR2CDK1
SCHEMBL241436 0.89 ADORA2A (0.41) ADORA2A
SCHEMBL4123170 0.89 ADORA2A (0.33) ADORA2ACDK1CDK5
SCHEMBL4119749 0.89 ADORA3 (0.34) ADORA2A
SCHEMBL4121510 0.88 ADORA2A (0.37) ADORA2A
SCHEMBL1402067 0.88 ADORA2A (0.38) ADORA2ACDK1CDK5
SCHEMBL4125460 0.88 CDK1 (0.32) ADORA2ACDK1CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2292619-A1 Purine derivatives for use as adenonsin A-2A receptor agonists Novartis AG (CH) 2011-03-09 EP disclosed