SCHEMBL14022752

SCHEMBL14022752

C=C(c1sc2ncn(CC(=O)N(CC)CC(F)(F)F)c(=O)c2c1C)N1CCN(c2ccc(C(F)(F)F)cc2)CC1

nearest known ligand 0.65

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
ALDH1A1 P00352 2/20 0.51
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
GAA P10253 1/20 0.51
SMN1; SMN2 Q16637 2/20 0.47
THRB P10828 1/20 0.41
TP53 P04637 1/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14022726 0.95 ALDH1A1 (0.56) CYP3A4CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL265880 0.93 CYP3A4 (0.62) CYP3A4CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL263878 0.88 CYP3A4 (0.65) CYP3A4CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL264374 0.85 CYP3A4 (0.61) CYP3A4CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL263727 0.81 CYP3A4 (0.55) CYP3A4CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL262628 0.79 MEN1 (0.56) CYP3A4CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL263410 0.78 CYP3A4 (0.66) CYP3A4CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL264526 0.77 CYP3A4 (0.65) CYP3A4CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL265919 0.77 CYP3A4 (0.58) CYP3A4CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL262985 0.74 SMN1; SMN2 (0.59) CYP3A4CYP2D6CYP2C9CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008138126-A1 BICYCLIC PYRIMIDINE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS NEUROMED PHARMACEUTICALS LTD. (CA) 2008-11-20 WO disclosed