SCHEMBL14025537

SCHEMBL14025537

CN(Cc1ccc(S(=O)(=O)N(C)Cc2ccccn2)cc1)C1CCCc2cccnc21

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 18/20 0.50
KCNH2 Q12809 1/20 0.45
PDE4A P27815 1/20 0.45
PDE4B Q07343 1/20 0.45
PDE4C Q08493 1/20 0.45
PDE4D Q08499 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
TAS2R14 Q9NYV8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14025523 0.85 CXCR4 (0.53) CXCR4KCNH2CYP3A4CYP2D6
SCHEMBL14025641 0.83 CXCR4 (0.49) CXCR4KCNH2
SCHEMBL14025539 0.81 CXCR4 (0.44) CXCR4KCNH2CYP2D6TAS2R14
SCHEMBL14025481 0.80 CXCR4 (0.48) CXCR4KCNH2
SCHEMBL14393283 0.78 CXCR4 (0.56) CXCR4KCNH2CYP2D6
SCHEMBL14025404 0.78 CXCR4 (0.58) CXCR4PDE4APDE4BPDE4CPDE4D
SCHEMBL21743932 0.77 CXCR4 (0.59) CXCR4KCNH2CYP3A4CYP2D6
SCHEMBL14025468 0.76 TAS2R14 (0.60) CXCR4PDE4APDE4BPDE4CPDE4D
SCHEMBL14025469 0.76 HDAC1 (0.56) CXCR4CYP3A4CYP2D6
SCHEMBL14025693 0.75 CXCR4 (0.51) CXCR4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080261978-A1 treating or preventing HIV infections, and in treating proliferative disorders such as inhibiting the metastasis of various cancers; 1-(4-((pyridin-2-ylmethylamino)methyl)benzyl)-3-phenylurea METASTATIX, INC. 2008-10-23 US disclosed
US-20080261978-A1 treating or preventing HIV infections, and in treating proliferative disorders such as inhibiting the metastasis of various cancers; 1-(4-((pyridin-2-ylmethylamino)methyl)benzyl)-3-phenylurea METASTATIX, INC. 2008-10-23 US disclosed
WO-2008109154-A1 CHEMOKINE RECEPTOR MODULATORS ALTIRIS THERAPEUTICS, INC. (US) 2008-09-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080261978-A1 treating or preventing HIV infections, and in treating proliferative disorders such as inhibiting the metastasis of various cancers; 1-(4-((pyridin-2-ylmethylamino)methyl)benzyl)-3-phenylurea MKI67, CCNI, CDKN1A CXCR4 242/4885KCNH2 3768/4885PDE4A 2435/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.