SCHEMBL14025569

SCHEMBL14025569

O=S(=O)(c1cccc(CNCc2ccccc2)c1)N(Cc1ccccc1)C1CCCc2cccnc21

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 15/20 0.47
CYP3A4 P08684 11/20 0.47
CYP2D6 P10635 11/20 0.47
TAS2R14 Q9NYV8 1/20 0.42
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
PSEN1 P49768 1/20 0.39
PSEN2 P49810 1/20 0.39
APH1B Q8WW43 1/20 0.39
NCSTN Q92542 1/20 0.39
APH1A Q96BI3 1/20 0.39
PSENEN Q9NZ42 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14025554 0.94 CXCR4 (0.53) CXCR4CYP3A4CYP2D6TAS2R14PDE4A
SCHEMBL14025404 0.86 CXCR4 (0.58) CXCR4CYP3A4CYP2D6TAS2R14PDE4A
SCHEMBL14025571 0.85 TAS2R14 (0.54) TAS2R14PDE4APDE4BPDE4CPDE4D
SCHEMBL14025556 0.84 PDE4A (0.52) CXCR4CYP3A4CYP2D6TAS2R14PDE4A
SCHEMBL14025587 0.83 CXCR4 (0.49) CXCR4CYP3A4CYP2D6
SCHEMBL14068398 0.82 TAS2R14 (0.47) CXCR4CYP3A4CYP2D6TAS2R14LMNA
SCHEMBL14025642 0.82 HDAC1 (0.48) CXCR4CYP3A4CYP2D6PDE4APDE4B
SCHEMBL14025641 0.80 CXCR4 (0.49) CXCR4
SCHEMBL14025607 0.79 TAS2R14 (0.48) TAS2R14PDE4APDE4BPDE4CPDE4D
SCHEMBL14025631 0.79 HDAC1 (0.49) CXCR4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080261978-A1 treating or preventing HIV infections, and in treating proliferative disorders such as inhibiting the metastasis of various cancers; 1-(4-((pyridin-2-ylmethylamino)methyl)benzyl)-3-phenylurea METASTATIX, INC. 2008-10-23 US disclosed
US-20080261978-A1 treating or preventing HIV infections, and in treating proliferative disorders such as inhibiting the metastasis of various cancers; 1-(4-((pyridin-2-ylmethylamino)methyl)benzyl)-3-phenylurea METASTATIX, INC. 2008-10-23 US disclosed
WO-2008109154-A1 CHEMOKINE RECEPTOR MODULATORS ALTIRIS THERAPEUTICS, INC. (US) 2008-09-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080261978-A1 treating or preventing HIV infections, and in treating proliferative disorders such as inhibiting the metastasis of various cancers; 1-(4-((pyridin-2-ylmethylamino)methyl)benzyl)-3-phenylurea MKI67, CCNI, CDKN1A CXCR4 242/4885CYP3A4 821/4885CYP2D6 962/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.