SCHEMBL14028515

SCHEMBL14028515

Oc1ccccc1-c1cc(C2CCCNC2)c2cn[nH]c2n1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 12/20 0.58
CHUK O15111 1/20 0.58
PRKCZ Q05513 1/20 0.43
PRKD2 Q9BZL6 1/20 0.43
CHEK2 O96017 3/20 0.41
CDK2 P24941 2/20 0.41
CDK1 P06493 1/20 0.41
SMYD2 Q9NRG4 1/20 0.40
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
CHEK1 O14757 1/20 0.39
CCNA2 P20248 1/20 0.39
CCNA1 P78396 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4945886 0.99 IKBKB (0.57) IKBKBCHUKPRKCZPRKD2CHEK2
SCHEMBL14028464 0.79 IKBKB (0.64) IKBKBCHUKCDK2CDK1
Hydrochloric Acid SCHEMBL4947782 0.78 IKBKB (0.63) IKBKBCHUKCDK2CDK1
SCHEMBL14046503 0.78 IKBKB (0.75) IKBKBCHUKCDK2CDK1
SCHEMBL14028482 0.76 IKBKB (0.56) IKBKBCHUKPRKCZPRKD2CHEK2
SCHEMBL14028511 0.76 IKBKB (0.72) IKBKBCHUK
Hydrochloric Acid SCHEMBL4942324 0.76 IKBKB (0.55) IKBKBCHUKPRKCZPRKD2CHEK2
SCHEMBL14028470 0.75 IKBKB (0.70) IKBKBCHUKCHEK2CDK2CDK1
Hydrochloric Acid SCHEMBL4947756 0.75 IKBKB (0.71) IKBKBCHUK
SCHEMBL14028498 0.75 IKBKB (0.56) IKBKBCHUKCHEK2CDK2CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7435743-B2 Pyridine derivatives BAYER AKTIENGESELLSCHAFT (DE) 2008-10-14 US disclosed
US-7435743-B2 Pyridine derivatives BAYER AKTIENGESELLSCHAFT (DE) 2008-10-14 US disclosed
EP-1326856-B1 PYRIDINE DERIVATIVES WITH IKB-KINASE (IKK-BETA) INHIBITING ACTIVITY BAYER HEALTHCARE AG (DE) 2007-12-19 EP disclosed
US-7232909-B2 Pyridine derivatives BAYER AKTIENGESELLSCHAFT (DE) 2007-06-19 US disclosed
US-7232909-B2 Pyridine derivatives BAYER AKTIENGESELLSCHAFT (DE) 2007-06-19 US disclosed