SCHEMBL14031876

SCHEMBL14031876

Cc1cc2nc(-c3[nH]nc4c3CCN(C(=O)Nc3ccccc3)C4)[nH]c2cc1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPSE Q9Y251 1/20 0.47
TRPV1 Q8NER1 10/20 0.42
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
POLB P06746 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 1/20 0.42
KDR P35968 1/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
TP53 P04637 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
THRB P10828 1/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
FAAH O00519 1/20 0.40
PDE10A Q9Y233 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14032076 0.91 HPSE (0.48) HPSETRPV1KDM4EMEN1CYP1A2
SCHEMBL14031950 0.91 NPC1 (0.46) HPSETRPV1KDM4EMEN1KMT2A
SCHEMBL14032114 0.90 SMN1; SMN2 (0.47) HPSETRPV1KDM4EKMT2ANPC1
SCHEMBL14032050 0.88 POLB (0.44) HPSETRPV1MEN1POLBKMT2A
SCHEMBL14032075 0.87 CYP1A2 (0.54) HPSETRPV1KDM4ECYP1A2CYP3A4
SCHEMBL14032053 0.86 MAPT (0.58) TRPV1KDM4EMEN1POLBKMT2A
SCHEMBL14031953 0.86 HPSE (0.40) HPSETRPV1KDM4EMEN1CYP1A2
SCHEMBL3457136 0.86 MTHFD2 (0.41) HPSETRPV1KDRNPC1RAB9A
SCHEMBL5067955 0.85 SMN1; SMN2 (0.45) HPSEKDM4ECYP1A2POLBCYP3A4
SCHEMBL14031928 0.85 HPSE (0.39) HPSEKDM4EMEN1CYP1A2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7435820-B2 Substituted tetrahydro-1H-pyrazolo [3,4-c]pyridines compositions comprising them, and use AVENTIS PHARMA S.A. (FR) 2008-10-14 US disclosed
US-7435820-B2 Substituted tetrahydro-1H-pyrazolo [3,4-c]pyridines compositions comprising them, and use AVENTIS PHARMA S.A. (FR) 2008-10-14 US disclosed