SCHEMBL14033593

SCHEMBL14033593

Clc1ccc(C(Cl)c2ccc(Br)cn2)cc1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 13/20 0.43
S1PR1 P21453 7/20 0.43
S1PR4 O95977 4/20 0.43
S1PR2 O95136 3/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CNR1 P21554 3/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
HIF1A Q16665 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14033306 1.00 S1PR3 (0.43) S1PR3S1PR1S1PR4S1PR2NPC1
SCHEMBL4602819 0.84 S1PR3 (0.43) S1PR3S1PR1S1PR4S1PR2MEN1
SCHEMBL14033749 0.84 S1PR3 (0.51) S1PR3S1PR4S1PR2NPC1RAB9A
SCHEMBL14033932 0.84 S1PR3 (0.51) S1PR3S1PR4S1PR2NPC1RAB9A
SCHEMBL23716350 0.81 S1PR3 (0.55) S1PR3S1PR1S1PR4S1PR2NPC1
SCHEMBL14033601 0.81 S1PR3 (0.45) S1PR3S1PR1S1PR4S1PR2NPC1
SCHEMBL14033902 0.80 TRPV1 (0.39) S1PR3S1PR1S1PR4S1PR2
SCHEMBL14033813 0.80 TRPV1 (0.39) S1PR3S1PR1S1PR4S1PR2
SCHEMBL4603195 0.77 S1PR3 (0.40) S1PR3S1PR1S1PR4S1PR2MEN1
SCHEMBL14585677 0.77 S1PR3 (0.40) S1PR3S1PR1S1PR4S1PR2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7432268-B2 17β-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases SCHERING CORPORATION (US) 2008-10-07 US disclosed
US-7432268-B2 17β-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases SCHERING CORPORATION (US) 2008-10-07 US disclosed