SCHEMBL1403369

SCHEMBL1403369

CC(=O)[CH]N

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28559756 0.96
Acetone SCHEMBL2428423 0.73
SCHEMBL306102 0.72
SCHEMBL28193228 0.72
SCHEMBL1843586 0.72
SCHEMBL12997105 0.72
Acetamide SCHEMBL6731735 0.70
Acetone SCHEMBL28344975 0.70 ALDH1A1 (0.53)
Acetic Acid SCHEMBL4942868 0.70 FFAR3 (0.58)
Acetic Acid SCHEMBL1342560 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 182 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106478841-B By being freeze-dried and the cysteine conjugates of hyaluronic acid of mercaptan-alkene clicking chemistry preparation and its synthetic method and application 海南大学 2019-02-19 CN claimed
CN-108148115-A A kind of cyclic peptide new synthetic method and its application in drug development 中国药科大学 2018-06-12 CN claimed
CN-106478841-A The cysteine conjugates of hyaluronic acid prepared with mercaptan alkene clicking chemistry by lyophilization and its synthetic method and application 海南大学 2017-03-08 CN claimed
CN-102844305-B Antibacterial isoquinolin-3-ylurea derivatives ACTELION PHARMACEUTICALS LTD 2014-07-02 CN claimed
CN-103429596-A Degradation of penicillin compounds DSM SINOCHEM PHARM NL BV 2013-12-04 CN claimed
CN-101693738-B Method for synthesizing terlipressin by solid-phase oxidization and cyclization SHENZHEN HYBIO PHARMACEUTICAL 2013-02-13 CN claimed
CN-102844305-A Antibacterial isoquinolin-3-ylurea derivatives ACTELION PHARMACEUTICALS LTD 2012-12-26 CN claimed
CN-102459160-A Lysine compounds and their use in site- and chemoselective modification of peptides and proteins STICHTING HET NL KANKER I 2012-05-16 CN claimed
CN-102112449-A Phenyl or pyridinyl substituted indazoles derivatives ASTRAZENECA AB 2011-06-29 CN claimed
CN-102037007-A Selective exosite inhibition of PAPP-A activity against IGFBP-4 UNIV AARHUS 2011-04-27 CN claimed
EP-2291359-A1 PHENYL OR PYRIDINYL SUBSTITUTED INDAZOLES DERIVATIVES AstraZeneca AB (SE) 2011-03-09 EP claimed
US-20100080786-A1 Phenyl or Pyridinyl Substituted Indazoles Derivatives ASTRAZENECA AB (SE) 2010-04-01 US claimed
WO-2009142569-A1 PHENYL OR PYRIDINYL SUBSTITUTED INDAZOLES DERIVATIVES ASTRAZENECA AB (SE) 2009-11-26 WO claimed
CN-1051547-C Beta-lactams derivative and its prep. and use HOFFMANN LA ROCHE (CH) 2000-04-19 CN claimed
CN-1132752-A Beta-lactam derivatives, process for their preparation and their use HOFFMANN LA ROCHE (CH) 1996-10-09 CN claimed
CN-1055925-A Pyridine derivate and preparation method thereof ICI PLC (GB) 1991-11-06 CN claimed
CN-86104835-A VASOPRESSIN ANTAGONISTS 1986-12-17 CN claimed
CN-117209447-A Compounds and compositions for treating disorders associated with NLRP activity 诺华股份有限公司 2023-12-12 CN disclosed
US-4857630-A Hyperbranched polyarylene E. I. DU PONT DE NEMOURS AND COMPANY (US) 1989-08-15 US disclosed
CN-86104835-A VASOPRESSIN ANTAGONISTS 1986-12-17 CN disclosed