SCHEMBL14035283

SCHEMBL14035283

CC(C)(C)OC(=O)N1CCN([C@H](CO)c2cccnc2)CC1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.58
CYP3A5 P20815 3/20 0.58
GPR119 Q8TDV5 1/20 0.51
PLA2G7 Q13093 1/20 0.51
MGLL Q99685 1/20 0.51
ABHD6 Q9BV23 1/20 0.51
TP53 P04637 2/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
HSD17B10 Q99714 1/20 0.47
NAMPT P43490 1/20 0.46
GBA1 P04062 1/20 0.46
TSHR P16473 1/20 0.46
MEN1 O00255 1/20 0.46
CYP2C19 P33261 1/20 0.46
KMT2A Q03164 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
POLB P06746 1/20 0.46
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20818634 0.91 CYP3A4 (0.58) CYP3A4CYP3A5GPR119PLA2G7MGLL
SCHEMBL30476445 0.91 CYP3A4 (0.58) CYP3A4CYP3A5GPR119PLA2G7MGLL
SCHEMBL31071488 0.86 CYP3A4 (0.71) CYP3A4CYP3A5GPR119PLA2G7MGLL
SCHEMBL15093706 0.86 CYP3A4 (0.71) CYP3A4CYP3A5GPR119PLA2G7MGLL
SCHEMBL5410711 0.86 ATM (0.50) GPR119MGLLKDM4EALDH1A1TSHR
SCHEMBL210120 0.85 CYP3A4 (0.61) CYP3A4CYP3A5GPR119PLA2G7MGLL
SCHEMBL29363322 0.83 CYP3A4 (0.59) CYP3A4CYP3A5GPR119PLA2G7MGLL
SCHEMBL19668681 0.83 CYP3A4 (0.59) CYP3A4CYP3A5GPR119PLA2G7MGLL
SCHEMBL8473520 0.80 CYP3A4 (0.53) CYP3A4CYP3A5GPR119PLA2G7MGLL
SCHEMBL8473516 0.80 CYP3A4 (0.53) CYP3A4CYP3A5GPR119PLA2G7MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008134036-A1 ALPHA-SUBSTITUTED ARYLMETHYL PIPERAZINE PYRAZOLO[1,5-α]PYRIMIDINE AMIDE DERIVATIVES PANACOS PHARMACEUTICALS, INC. (US) 2008-11-06 WO disclosed