SCHEMBL14039059

SCHEMBL14039059

CC(C)(C)NC(=O)Nc1nc2nc(O)ncc2cc1Oc1ccc(F)cc1F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 17/20 0.48
PDGFRB P09619 14/20 0.48
PDGFRA P16234 14/20 0.48
SRC P12931 12/20 0.48
EGFR P00533 4/20 0.43
FGFR2 P21802 4/20 0.43
FGFR4 P22455 4/20 0.43
FGFR3 P22607 4/20 0.43
MAPK14 Q16539 2/20 0.43
MAPK8 P45983 1/20 0.41
PRKD3 O94806 1/20 0.41
PRKCG P05129 1/20 0.41
PRKCB P05771 1/20 0.41
PRKCA P17252 1/20 0.41
PRKCH P24723 1/20 0.41
MAPK3 P27361 1/20 0.41
MAPK1 P28482 1/20 0.41
PRKCI P41743 1/20 0.41
PRKCE Q02156 1/20 0.41
PRKCQ Q04759 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5111814 0.88 FGFR1 (0.46) FGFR1PDGFRBPDGFRASRCEGFR
SCHEMBL5114782 0.87 FGFR1 (0.45) FGFR1PDGFRBPDGFRASRCEGFR
SCHEMBL5107303 0.81 MAPK14 (0.57) MAPK14MAPK8PRKD3MAPK1
SCHEMBL29594951 0.81 MAPK14 (0.57) MAPK14MAPK8PRKD3MAPK1
SCHEMBL13530692 0.71 FGFR1 (0.45) FGFR1PDGFRBPDGFRASRCEGFR
SCHEMBL5122174 0.66 MAPK8 (0.43) MAPK14MAPK8
SCHEMBL25222319 0.65 MAPK8 (0.42) MAPK14MAPK8
SCHEMBL29536776 0.65 MAPK8 (0.42) MAPK14MAPK8
SCHEMBL6073910 0.65 FGFR1 (0.50) FGFR1PDGFRBPDGFRASRCEGFR
SCHEMBL8129964 0.65 FGFR1 (1.00) FGFR1PDGFRBPDGFRASRCEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7449581-B2 6-Substituted pyrido-pyrimidines POCHE PALO ALTO LLC (US) 2008-11-11 US disclosed