SCHEMBL14040985

SCHEMBL14040985

O=C(Cl)c1cccnc1Sc1ccc(Cl)cc1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.58
KDM4E B2RXH2 2/20 0.58
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2C9 P11712 1/20 0.58
HPGD P15428 1/20 0.58
CYP2C19 P33261 1/20 0.58
SMN1; SMN2 Q16637 3/20 0.55
MEN1 O00255 3/20 0.55
KMT2A Q03164 3/20 0.55
GAA P10253 1/20 0.55
LMNA P02545 1/20 0.54
NPC1 O15118 1/20 0.48
PKM P14618 1/20 0.48
L3MBTL1 Q9Y468 2/20 0.47
ATM Q13315 1/20 0.47
CRHBP P24387 1/20 0.46
CRHR2 Q13324 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
MAPT P10636 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7108755 0.88 ALDH1A1 (0.71) ALDH1A1KDM4ECYP1A2CYP3A4CYP2C9
SCHEMBL7110016 0.87 SMN1; SMN2 (0.61) ALDH1A1CYP2C9SMN1; SMN2MEN1KMT2A
SCHEMBL31544568 0.86 ALDH1A1 (0.74) ALDH1A1KDM4ECYP1A2CYP3A4HPGD
SCHEMBL4768446 0.86 ALDH1A1 (0.74) ALDH1A1KDM4ECYP1A2CYP3A4HPGD
SCHEMBL14040903 0.82 ALDH1A1 (0.53) ALDH1A1KDM4ECYP1A2CYP3A4CYP2C9
SCHEMBL14502540 0.78 ALDH1A1 (0.54) ALDH1A1KDM4ECYP1A2CYP3A4CYP2C9
SCHEMBL1514453 0.78 ALDH1A1 (0.67) ALDH1A1KDM4ECYP1A2CYP3A4CYP2C9
SCHEMBL4452821 0.78 SMN1; SMN2 (0.46) ALDH1A1KDM4ECYP3A4CYP2C9SMN1; SMN2
SCHEMBL8125018 0.77 ALDH1A1 (0.65) ALDH1A1KDM4ECYP1A2CYP3A4CYP2C9
SCHEMBL934289 0.75 KMT2A (0.56) ALDH1A1HPGDMEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539693-B9 CANNABINOID RECEPTOR AGONISTS SCHERING CORP (US) 2008-10-08 EP disclosed
EP-1539693-B1 CANNABINOID RECEPTOR AGONISTS SCHERING CORP (US) 2008-03-12 EP disclosed
US-7217732-B2 Cannabinoid receptor agonists SCHERING CORPORATION (US) 2007-05-15 US disclosed
US-7217732-B2 Cannabinoid receptor agonists SCHERING CORPORATION (US) 2007-05-15 US disclosed