SCHEMBL14045239

SCHEMBL14045239

CN(C1CCN(CC(F)(F)F)CC1)S(=O)(=O)c1ccc(N)cc1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 17/20 0.56
HTR2C P28335 13/20 0.56
L3MBTL1 Q9Y468 3/20 0.49
ALDH1A1 P00352 2/20 0.47
GAA P10253 2/20 0.47
HTR1A P08908 3/20 0.47
DRD2 P14416 3/20 0.47
HTR7 P34969 3/20 0.47
DPP4 P27487 1/20 0.46
DPP8 Q6V1X1 1/20 0.46
DPP9 Q86TI2 1/20 0.46
DPP7 Q9UHL4 1/20 0.46
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14045127 0.88 HTR2A (0.57) HTR2AHTR2CL3MBTL1ALDH1A1GAA
SCHEMBL14045062 0.86 HTR2A (0.52) HTR2AHTR2CL3MBTL1ALDH1A1GAA
SCHEMBL14045199 0.86 HTR2A (0.55) HTR2AHTR2CL3MBTL1ALDH1A1GAA
SCHEMBL14045067 0.82 CACNA1B (0.39) HTR2AHTR2CALDH1A1HTR1ADRD2
SCHEMBL14045243 0.81 HTR2A (0.54) HTR2AHTR2CL3MBTL1ALDH1A1GAA
SCHEMBL14625133 0.81 HTR2A (0.57) HTR2AHTR2CL3MBTL1ALDH1A1GAA
SCHEMBL14625270 0.80 HTR2A (0.76) HTR2AHTR2CL3MBTL1ALDH1A1GAA
SCHEMBL14045248 0.80 HTR2A (0.62) HTR2AHTR2CL3MBTL1HTR1ADRD2
SCHEMBL27895777 0.79 ALDH1A1 (0.57) HTR2AHTR2CL3MBTL1ALDH1A1GAA
SCHEMBL14045250 0.79 HTR2A (0.58) HTR2AHTR2CL3MBTL1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080269170-A1 Novel 2,4-Dianilinopyrimidine Derivatives, the Preparation Thereof, Their Use as Medicaments, Pharmaceutical Compositions and, in Particular, as IKK Inhibitors SANOFI-AVENTIS (FR) 2008-10-30 US disclosed
WO-2007006926-A2 NOVEL 2,4-DIANILINOPYRIMIDINE DERIVATIVES, THE PREPARATION THEREOF, THEIR USE AS MEDICAMENTS, PHARMACEUTICAL COMPOSITIONS AND, IN PARTICULAR, AS IKK INHIBITORS SANOFI-AVENTIS (FR) 2007-01-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080269170-A1 Novel 2,4-Dianilinopyrimidine Derivatives, the Preparation Thereof, Their Use as Medicaments, Pharmaceutical Compositions and, in Particular, as IKK Inhibitors NFKBIA, IKBKB, IKBKE HTR2A 3453/4885HTR2C 3934/4885L3MBTL1 4039/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.