SCHEMBL14045940

SCHEMBL14045940

CCc1ccc2cc(CF)ccc2n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TERT O14746 1/20 0.38
CYP1A2 P05177 2/20 0.37
CYP2A6 P11509 1/20 0.37
PDE10A Q9Y233 3/20 0.35
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
MEN1 O00255 2/20 0.35
ALDH1A1 P00352 2/20 0.35
KMT2A Q03164 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
ADORA2A P29274 1/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
HPGD P15428 1/20 0.35
PTK2B Q14289 1/20 0.35
KDM4E B2RXH2 1/20 0.33
TSHR P16473 1/20 0.33
CASP1 P29466 1/20 0.33
GRM1 Q13255 1/20 0.33
DHFR P00374 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12824284 0.87 CYP1A2 (0.50) TERTCYP1A2CYP2A6PDE10ANPC1
SCHEMBL7837249 0.82 NPC1 (0.38) TERTCYP1A2CYP2A6NPC1RAB9A
SCHEMBL9697024 0.82 CYSLTR1 (0.42) TERTCYP1A2CYP2A6PDE10ANPC1
SCHEMBL18949111 0.79 ADORA2A (0.36) TERTCYP1A2CYP2A6PDE10ANPC1
SCHEMBL24060260 0.78 PDE10A (0.51) CYP1A2PDE10ANPC1RAB9ALMNA
SCHEMBL25728354 0.78 HRH3 (0.43) TERT
SCHEMBL7838005 0.78 BACE1 (0.53) TERTCYP1A2CYP2A6PDE10AMEN1
SCHEMBL6230105 0.76 CYP1A2 (0.59) CYP1A2CYP2A6NPC1RAB9AMEN1
SCHEMBL7813726 0.75 CYP1A2 (0.46) CYP1A2CYP2A6NPC1RAB9AMEN1
SCHEMBL5050008 0.74 BACE1 (0.53) TERTCYP1A2CYP2A6MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8323621-B2 site-directed delivery of contrast agent; brain or breast cancer; 1,4,7,10 tetraazacyclododecane having variable chelating ions, phosphoester chains, and light harvesting moieties for changing imaging methods; conjugated to high affinity PBR ligand PK11195; bound to a PVA or a PEG delivery vehicle VANDERBILT UNIVERSITY (US) 2012-12-04 US disclosed
US-20080241074-A1 MULTI-USE MULTIMODAL IMAGING CHELATES VANDERBILT UNIVERSITY 2008-10-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080241074-A1 MULTI-USE MULTIMODAL IMAGING CHELATES PCNA, CLTC, CLTB TERT 3946/4885CYP1A2 4559/4885CYP2A6 4458/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.