SCHEMBL14047840

SCHEMBL14047840

Nc1nc2c(c(=O)n1C(c1ccccc1)c1ccccc1)CCNC2

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 8/20 0.39
PARP1 P09874 1/20 0.36
TNKS2 Q9H2K2 1/20 0.36
PARP2 Q9UGN5 1/20 0.36
HTR2C P28335 6/20 0.34
HTR2B P41595 3/20 0.34
HTR2A P28223 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
F12 P00748 2/20 0.33
HTR6 P50406 1/20 0.33
CD44 P16070 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14047930 0.93 HTR2A (0.42) SIGMAR1HTR2CHTR2BHTR2A
SCHEMBL13329622 0.90 HTR2C (0.37) SIGMAR1PARP1TNKS2HTR2CHTR2B
SCHEMBL14047939 0.88 SIGMAR1 (0.41) SIGMAR1PARP1TNKS2PARP2HTR2C
SCHEMBL13249768 0.85 SIGMAR1 (0.41) SIGMAR1PARP1TNKS2PARP2HTR2C
SCHEMBL14047692 0.83 SIGMAR1 (0.35) SIGMAR1PARP1TNKS2PARP2HTR2C
SCHEMBL13250502 0.82 SIGMAR1 (0.39) SIGMAR1PARP1TNKS2PARP2HTR2C
SCHEMBL13250510 0.82 SIGMAR1 (0.39) SIGMAR1PARP1TNKS2PARP2HTR2C
SCHEMBL13250516 0.79 SIGMAR1 (0.36) SIGMAR1PARP1TNKS2PARP2HTR2C
SCHEMBL14047934 0.77 HTR2A (0.31) HTR2AMEN1KMT2A
SCHEMBL13250488 0.77 HTR2A (0.32) HTR2AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008130581-A1 PYRIMIDINONE DERIVATIVES AND METHODS OF USE THEREOF SCHERING CORPORATION (US) 2008-10-30 WO disclosed