SCHEMBL14048441

SCHEMBL14048441

Cc1csc2cc(C(C)(F)F)ccc12

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.41
CYP17A1 P05093 1/20 0.32
KIF11 P52732 1/20 0.32
CHRNA7 P36544 1/20 0.31
HTR3A P46098 1/20 0.31
PPARG P37231 1/20 0.31
PPARD Q03181 1/20 0.31
PPARA Q07869 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL699328 0.87 CYP2A6 (0.42) CYP2A6KIF11PPARGPPARDPPARA
SCHEMBL26144297 0.85 CYP2A6 (0.43) CYP2A6CYP17A1KIF11CHRNA7HTR3A
SCHEMBL2095399 0.73 CYP2A6 (0.46) CYP2A6KIF11
SCHEMBL3684920 0.73 CYP2A6 (0.55) CYP2A6KIF11MEN1KMT2A
SCHEMBL424317 0.72 CYP2A6 (0.48) CYP2A6CYP17A1CHRNA7HTR3A
SCHEMBL5542590 0.72 NPC1 (0.42) CYP2A6KIF11
SCHEMBL13447302 0.72 HRH4 (0.36) KIF11PPARA
SCHEMBL25037436 0.70 CYP2A6 (0.56) CYP2A6KIF11CHRNA7HTR3AMEN1
SCHEMBL14093011 0.70 KIF11 (0.45) CYP17A1KIF11PPARGPPARDPPARA
SCHEMBL14048577 0.70 POLB (0.48) CYP2A6KIF11MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1632483-B1 HETEROCYCLIC SUBSTITUTED CARBONYL DERIVATIVES AND THEIR USE AS DOPAMINE D3 RECEPTOR LIGANDS AVENTIS PHARMA INC (US) 2008-10-29 EP disclosed