SCHEMBL14048620

SCHEMBL14048620

CNCCc1sc(N)nc1CF

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.37
HRH2 P25021 1/20 0.37
HRH1 P35367 1/20 0.37
HRH4 Q9H3N8 1/20 0.37
HTT P42858 1/20 0.33
ALDH1A1 P00352 1/20 0.30
GAA P10253 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13202887 0.77 HRH2 (0.63) CYP1A2HRH2HRH1HRH4ALDH1A1
SCHEMBL31612254 0.67 HRH2 (0.59) CYP1A2HRH2HRH1HRH4
SCHEMBL8259817 0.67 ALDH1A1 (0.41) CYP1A2HRH2HRH1HRH4HTT
SCHEMBL10986689 0.64 ALDH1A1 (0.49) CYP1A2HRH2HRH1HRH4HTT
SCHEMBL13459260 0.63
SCHEMBL2175079 0.61 ALDH1A1 (0.48) CYP1A2HRH2HRH1HRH4HTT
SCHEMBL24202463 0.61 ALDH1A1 (0.50) CYP1A2HRH2HRH1HRH4ALDH1A1
SCHEMBL31612250 0.60 HRH2 (0.59) CYP1A2HRH2HRH1HRH4HTT
Hydrochloric Acid SCHEMBL10987975 0.59 ALDH1A1 (0.47) CYP1A2HRH2HRH1HRH4HTT
SCHEMBL31612261 0.59 HRH2 (0.58) CYP1A2HRH2HRH1HRH4HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1632483-B1 HETEROCYCLIC SUBSTITUTED CARBONYL DERIVATIVES AND THEIR USE AS DOPAMINE D3 RECEPTOR LIGANDS AVENTIS PHARMA INC (US) 2008-10-29 EP disclosed