SCHEMBL14049280

SCHEMBL14049280

COC(=O)CC(=O)Nc1ccccc1S(N)(=O)=O

nearest known ligand 0.68

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CA1 P00915 19/20 0.68
CA2 P00918 19/20 0.68
CA4 P22748 2/20 0.54
CA9 Q16790 3/20 0.51
CA5A P35218 1/20 0.50
CA12 O43570 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL392166 0.87 CA1 (0.62) CA1CA2CA4CA9CA12
SCHEMBL8760294 0.84 CA1 (0.77) CA1CA2CA4CA9CA12
SCHEMBL15873682 0.81 CA1 (0.45) CA1CA2CA4CA9CA5A
SCHEMBL14338090 0.81 MEN1 (0.49) CA1CA2CA4CA9CA5A
SCHEMBL7481802 0.81 CA1 (0.61) CA1CA2CA9CA5ACA12
SCHEMBL13686435 0.80 CA1 (0.44) CA1CA2CA4CA9CA5A
SCHEMBL7492311 0.80 CA1 (0.69) CA1CA2CA4CA9CA12
SCHEMBL9023668 0.80 CA1 (0.56) CA1CA2CA9CA5ACA12
SCHEMBL7933999 0.80 CA1 (0.73) CA1CA2CA4CA9CA5A
SCHEMBL5348269 0.78 ALDH1A1 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2129224-B1 5,6-DIHYDRO-1H-PYRIDIN-2-ONE COMPOUNDS ANADYS PHARMACEUTICALS INC (US) 2016-03-30 EP disclosed
US-20140031346-A1 5,6-DIHYDRO-1H-PYRIDIN-2-ONE COMPOUNDS ANADYS PHARMACEUTICALS, INC. (US) 2014-01-30 US disclosed
WO-2008124450-A1 5,6-DIHYDRO-1H-PYRIDIN-2-ONE COMPOUNDS ANADYS PHARMACEUTICALS, INC. (US) 2008-10-16 WO disclosed
WO-2008073982-A2 5,6-DIHYDRO-1H-PYRIDIN-2-ONE COMPOUNDS ANADYS PHARMACEUTICALS, INC. (US) 2008-06-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140031346-A1 5,6-DIHYDRO-1H-PYRIDIN-2-ONE COMPOUNDS HAVCR2, CCR3, C5 CA1 3513/4885CA2 3451/4885CA4 1792/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.