SCHEMBL14064871

SCHEMBL14064871

CC(C)CNC(C)(C)c1cnc(Nc2ccc(Cl)cc2Cl)cc1C(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 13/20 0.46
CYP2C9 P11712 3/20 0.46
CYP2C19 P33261 3/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2D6 P10635 2/20 0.46
CNR1 P21554 1/20 0.40
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
ALOX12 P18054 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
MAPK1 P28482 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.33
SRC P12931 1/20 0.33
TTK P33981 1/20 0.33
SCN1A P35498 1/20 0.32
SCN5A Q14524 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4649764 0.78 CNR2 (0.47) CNR2CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL14381958 0.75 CNR2 (0.56) CNR2CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL4649725 0.75 CNR2 (0.71) CNR2CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL4649722 0.75 CNR2 (0.52) CNR2CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL4648499 0.73 CNR2 (0.51) CNR2CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL4649620 0.71 CNR2 (0.62) CNR2CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL5213108 0.69 CNR2 (0.69) CNR2CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL14006020 0.67 CNR2 (0.46) CNR2CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL4649692 0.67 CNR2 (0.50) CNR2CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL4649694 0.67 CNR2 (0.58) CNR2CYP2C9CYP2C19CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1718613-B1 PYRIDINE DERIVATIVES AND THEIR USE AS CB2 RECEPTOR MODULATORS GLAXO GROUP LTD (GB) 2008-09-03 EP disclosed