SCHEMBL4649692

SCHEMBL4649692

CC(C)c1cc(Nc2ccc(Cl)cc2Cl)ncc1CN(C)C1CCC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 8/20 0.50
CYP2C9 P11712 3/20 0.50
CYP2C19 P33261 3/20 0.50
CYP1A2 P05177 2/20 0.50
CYP3A4 P08684 2/20 0.50
CYP2D6 P10635 2/20 0.50
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
CNR1 P21554 1/20 0.38
NOS3 P29474 7/20 0.38
NOS1 P29475 7/20 0.38
NOS2 P35228 7/20 0.38
CHEK1 O14757 1/20 0.37
NTRK1 P04629 1/20 0.37
FYN P06241 1/20 0.37
RET P07949 1/20 0.37
MET P08581 1/20 0.37
PDGFRB P09619 1/20 0.37
PIM1 P11309 1/20 0.37
FGFR1 P11362 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4649624 0.92 CNR2 (0.42) CNR2CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL4649775 0.82 CNR2 (0.40) CNR2CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL4649736 0.82 CDK4 (0.38) CNR2CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL4649694 0.81 CNR2 (0.58) CNR2CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL4649722 0.79 CNR2 (0.52) CNR2CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL4649780 0.77 CNR2 (0.37) CNR2CYP3A4CYP2D6CHEK1NTRK1
SCHEMBL4649712 0.77 CNR2 (0.54) CNR2NOS3NOS1NOS2ALDH1A1
SCHEMBL4649631 0.76 CNR2 (0.56) CNR2RAB9ACDK5POLB
SCHEMBL4649764 0.75 CNR2 (0.47) CNR2CYP2C9CYP2C19CYP1A2CYP3A4
SCHEMBL4649071 0.75 CNR2 (0.37) CNR2CYP2C9CYP2C19CYP1A2FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1718613-B1 PYRIDINE DERIVATIVES AND THEIR USE AS CB2 RECEPTOR MODULATORS GLAXO GROUP LTD (GB) 2008-09-03 EP disclosed