SCHEMBL14065014

SCHEMBL14065014

CC[C@H](CC#N)OC(C)=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
LMNA P02545 2/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
HRH1 P35367 1/20 0.35
KMT2A Q03164 1/20 0.35
SLC18A3 Q16572 1/20 0.34
PRKCA P17252 2/20 0.33
IMPDH2 P12268 1/20 0.33
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
CHRM1 P11229 1/20 0.32
TBXA2R P21731 1/20 0.32
GALR3 O60755 1/20 0.31
MAPT P10636 1/20 0.31
BLM P54132 1/20 0.31
CTSL P07711 1/20 0.31
CTSB P07858 1/20 0.31
CTSK P43235 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5580290 1.00 TSHR (0.36) TSHRSMN1; SMN2LMNAMEN1CYP1A2
SCHEMBL5580073 1.00 TSHR (0.36) TSHRSMN1; SMN2LMNAMEN1CYP1A2
SCHEMBL19493385 0.83 PRKCA (0.40) TSHRSMN1; SMN2LMNAMEN1CYP1A2
SCHEMBL7723645 0.82 AR (0.35) TSHRSMN1; SMN2LMNAMEN1CYP1A2
SCHEMBL7719955 0.82 AR (0.35) TSHRSMN1; SMN2LMNAMEN1CYP1A2
SCHEMBL7716828 0.82 AR (0.35) TSHRSMN1; SMN2LMNAMEN1CYP1A2
SCHEMBL13491728 0.80 TDP1 (0.44) TSHRSMN1; SMN2LMNAMEN1CYP1A2
SCHEMBL28797081 0.80 MAPT (0.34) PRKCAIMPDH2MAPTCTSLCTSB
SCHEMBL28797083 0.80 MAPT (0.34) PRKCAIMPDH2MAPTCTSLCTSB
SCHEMBL1584634 0.79

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1964561-A1 Inhibitors of IMPDH enzyme Vertex Pharmaceuticals Incorporated (US) 2008-09-03 EP disclosed