SCHEMBL14065145

SCHEMBL14065145

CNCCC(OC(=O)NCc1ccccc1)c1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
UTS2R Q9UKP6 1/20 0.60
CYP19A1 P11511 1/20 0.60
PPARG P37231 1/20 0.57
PPARA Q07869 1/20 0.57
SLC6A4 P31645 10/20 0.51
SLC6A2 P23975 6/20 0.47
CYP1A2 P05177 4/20 0.47
CYP3A4 P08684 4/20 0.47
CYP2D6 P10635 4/20 0.47
TSHR P16473 3/20 0.47
SLC6A3 Q01959 3/20 0.47
KMT2A Q03164 2/20 0.47
CHRM1 P11229 2/20 0.47
ADRA2B P18089 2/20 0.47
HTR2A P28223 2/20 0.47
HTR2C P28335 2/20 0.47
HRH1 P35367 2/20 0.47
OPRM1 P35372 2/20 0.47
DRD3 P35462 2/20 0.47
OPRK1 P41145 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14065176 0.83 UTS2R (0.84) UTS2RCYP19A1PPARGPPARA
SCHEMBL14064826 0.81 UTS2R (0.66) UTS2RCYP19A1PPARGPPARACYP1A2
SCHEMBL3277857 0.80 SLC6A4 (0.59) SLC6A4SLC6A2CYP1A2CYP3A4CYP2D6
SCHEMBL14065228 0.80 UTS2R (0.68) UTS2RCYP19A1PPARGPPARA
SCHEMBL14064819 0.79 SLC6A4 (0.58) SLC6A4SLC6A2CYP1A2CYP3A4CYP2D6
SCHEMBL21118559 0.78 TP53 (0.57) SLC6A4SLC6A2CYP1A2CYP3A4CYP2D6
SCHEMBL8077913 0.76 PPARG (0.53) UTS2RCYP19A1PPARGPPARAKMT2A
SCHEMBL27999195 0.76 CYP19A1 (0.61) UTS2RCYP19A1PPARGPPARACYP3A4
SCHEMBL20917307 0.76 SLC6A4 (0.59) SLC6A4SLC6A2KMT2A
SCHEMBL5455926 0.75 UTS2R (1.00) UTS2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1964561-A1 Inhibitors of IMPDH enzyme Vertex Pharmaceuticals Incorporated (US) 2008-09-03 EP disclosed