SCHEMBL14067374

SCHEMBL14067374

Cc1cc(I)nn2cc(-c3ccc(N(C)C)nc3)nc12

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
APP P05067 5/20 0.40
CRHR1 P34998 2/20 0.38
PSD A5PKW4 1/20 0.36
MAP3K11 Q16584 1/20 0.36
HPGD P15428 1/20 0.35
NPC1 O15118 1/20 0.35
POLB P06746 1/20 0.35
GAA P10253 1/20 0.35
RAB9A P51151 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
SYK P43405 3/20 0.35
TDO2 P48775 1/20 0.34
MAPT P10636 1/20 0.34
AURKB Q96GD4 1/20 0.34
ICMT O60725 1/20 0.34
PIK3CA P42336 1/20 0.34
MET P08581 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14067376 0.85 APP (0.39) APPCRHR1PSDHPGDNPC1
SCHEMBL14067306 0.82 APP (0.51) APPHPGDNPC1GAARAB9A
SCHEMBL14067384 0.79 APP (0.43) APPCRHR1PSDMAP3K11HPGD
SCHEMBL14067566 0.79 APP (0.40) APPMAP3K11HPGDNPC1POLB
SCHEMBL14067373 0.78 MAP3K11 (0.38) APPCRHR1MAP3K11HPGDNPC1
SCHEMBL14067385 0.74 NPC1 (0.44) APPCRHR1PSDHPGDNPC1
SCHEMBL14067408 0.73 APP (0.40) APPMAP3K11HPGDNPC1POLB
SCHEMBL14067371 0.73 APP (0.39) APPCRHR1PSDMAP3K11HPGD
SCHEMBL14067318 0.72 APP (0.31) APPNPC1RAB9A
SCHEMBL14067382 0.72 APP (0.43) APPNPC1RAB9ASYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080219922-A1 Alzheimer's Disease Imaging Agents EMORY UNIVERSITY 2008-09-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080219922-A1 Alzheimer's Disease Imaging Agents APP, PSEN1, MAPT APP 1/4885CRHR1 2786/4885PSD 489/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.