SCHEMBL14067971

SCHEMBL14067971

CCOC(=O)CCn1c2c(c3cc(C)ccc31)CNCC2

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 5/20 0.54
SIRT1 Q96EB6 3/20 0.52
HSD17B10 Q99714 2/20 0.47
CYP3A4 P08684 1/20 0.43
CNR2 P34972 2/20 0.42
HRH1 P35367 3/20 0.40
HTR6 P50406 3/20 0.40
ADRA2A P08913 2/20 0.40
HTR2A P28223 2/20 0.40
HTR2C P28335 2/20 0.40
HTR7 P34969 2/20 0.40
ADRA1A P35348 2/20 0.40
KDM4E B2RXH2 2/20 0.40
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.39
DRD2 P14416 1/20 0.39
POLB P06746 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
HDAC1 Q13547 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14216298 0.94 HSD17B10 (0.51) SIRT2SIRT1HSD17B10CYP3A4CNR2
SCHEMBL14067973 0.90 CYP3A4 (0.56) SIRT2SIRT1CYP3A4CNR2HRH1
SCHEMBL14067842 0.89 HSD17B10 (0.57) SIRT2SIRT1HSD17B10CYP3A4KDM4E
SCHEMBL14067969 0.87 KDM4E (0.53) SIRT2SIRT1CNR2HTR2AHTR2C
SCHEMBL10154872 0.83 HSD17B10 (0.61) SIRT2SIRT1HSD17B10KDM4EPTGDR2
SCHEMBL16140207 0.82 SIRT2 (0.59) SIRT2SIRT1HSD17B10CYP3A4HRH1
SCHEMBL3318769 0.82 HTR6 (0.62) SIRT2SIRT1HRH1HTR6ADRA2A
SCHEMBL16140204 0.80 SIRT2 (0.60) SIRT2SIRT1HSD17B10CYP3A4HRH1
SCHEMBL10127820 0.80 HRH1 (0.54) SIRT2SIRT1HSD17B10CNR2HRH1
SCHEMBL1120682 0.80 HRH1 (0.51) HSD17B10CNR2HRH1HTR6ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008115098-A2 SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-PYRIDO[4,3-B]INDOLES, METHODS FOR THE PRODUCTION AND THE USE THEREOF ALLA CHEM, LLC (US) 2008-09-25 WO disclosed