SCHEMBL14068604

SCHEMBL14068604

Cc1cncc(Nc2ccc(CO)cc2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.42
XDH P47989 3/20 0.40
SLC22A12 Q96S37 3/20 0.40
FPR2 P25090 1/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
GRM4 Q14833 1/20 0.39
BRAF P15056 1/20 0.38
ATM Q13315 1/20 0.38
HCAR2 Q8TDS4 1/20 0.37
MEN1 O00255 1/20 0.36
GAA P10253 1/20 0.36
G6PD P11413 1/20 0.36
KMT2A Q03164 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CYP2A6 P11509 1/20 0.36
TYR P14679 1/20 0.35
PIK3CA P42336 1/20 0.35
SYK P43405 1/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14031002 0.82 XDH (0.48) PDPK1XDHSLC22A12BRAFMEN1
SCHEMBL14005509 0.80 XDH (0.43) PDPK1XDHSLC22A12BRAFTYR
SCHEMBL22042452 0.80 PDPK1 (0.47) PDPK1XDHSLC22A12CHRNB4CHRNA3
SCHEMBL14409688 0.78 HPGD (0.54) MEN1GAAG6PDKMT2AL3MBTL1
SCHEMBL5462060 0.76 NPSR1 (0.63) MEN1GAAKMT2AL3MBTL1NPC1
SCHEMBL4187435 0.74 XDH (0.56) PDPK1XDHSLC22A12CHRNB4CHRNA3
SCHEMBL13743490 0.74 MKNK1 (0.53) BRAFHCAR2CYP2A6
SCHEMBL13169061 0.73 TSHR (0.42) MEN1GAAG6PDKMT2AL3MBTL1
SCHEMBL14031014 0.73 SCN10A (0.45) CHRNB4CHRNA3GRM4CYP2A6SYK
SCHEMBL1630903 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008109613-A1 BENZO[C][2,7]NAPHTHYRIDINE DERIVATIVES, AND THEIR USE AS KINASE INHIBITORS WYETH (US) 2008-09-12 WO disclosed