SCHEMBL14069237

SCHEMBL14069237

CNC(=O)[C@@H]1C[C@@H](OC(C)(C)OC)[C@H](n2cnc3c(NCc4cccc(I)c4)ncnc32)O1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 10/20 0.64
ADORA2A P29274 4/20 0.64
ADORA1 P30542 3/20 0.64
CYP3A4 P08684 2/20 0.64
MAPK1 P28482 2/20 0.64
CYP1A2 P05177 1/20 0.64
MAPT P10636 1/20 0.64
LMNA P02545 1/20 0.64
BLM P54132 1/20 0.64
PMP22 Q01453 1/20 0.64
CYP2D6 P10635 1/20 0.64
PKM P14618 1/20 0.64
TSHR P16473 1/20 0.64
NFKB1 P19838 1/20 0.64
ABCG2 Q9UNQ0 1/20 0.64
HTR2C P28335 1/20 0.64
ADORA2B P29275 1/20 0.64
HTR2B P41595 1/20 0.64
RXFP1 Q9HBX9 1/20 0.64
PPARD Q03181 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13456378 0.83 ADORA3 (0.67) ADORA3ADORA2AADORA1CYP3A4MAPK1
SCHEMBL24601177 0.80 ADORA3 (0.68) ADORA3ADORA2AADORA1CYP3A4MAPK1
SCHEMBL13400311 0.80 ADORA3 (0.69) ADORA3ADORA2AADORA1CYP3A4MAPK1
Ib-Meca SCHEMBL448115 0.78 ADORA3 (1.00) ADORA3ADORA2AADORA1CYP3A4MAPK1
Ib-Meca SCHEMBL465039 0.78 ADORA3 (1.00) ADORA3ADORA2AADORA1CYP3A4MAPK1
Ib-Meca SCHEMBL29634441 0.78 ADORA3 (1.00) ADORA3ADORA2AADORA1CYP3A4MAPK1
Ib-Meca SCHEMBL8922766 0.78 ADORA3 (1.00) ADORA3ADORA2AADORA1CYP3A4MAPK1
Ib-Meca SCHEMBL10089244 0.78 ADORA3 (1.00) ADORA3ADORA2AADORA1CYP3A4MAPK1
Ib-Meca SCHEMBL20905217 0.78 ADORA3 (1.00) ADORA3ADORA2AADORA1CYP3A4MAPK1
Ib-Meca SCHEMBL10089200 0.78 ADORA3 (1.00) ADORA3ADORA2AADORA1CYP3A4MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008111082-A1 PROCESS FOR THE SYNTHESIS OF IB-MECA CAN-FITE BIOPHARMA LTD. (IL) 2008-09-18 WO disclosed