SCHEMBL14075397

SCHEMBL14075397

COC(=O)c1cccc(Oc2ccc(NS(=O)(=O)c3ccc([N+](=O)[O-])cc3)c(C(=O)O)c2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 4/20 0.60
CYP1A2 P05177 1/20 0.60
KMT2A Q03164 3/20 0.58
MEN1 O00255 2/20 0.58
KDM4E B2RXH2 2/20 0.55
ALDH1A1 P00352 3/20 0.52
PYGL P06737 1/20 0.51
CYP2C19 P33261 1/20 0.50
MAPT P10636 2/20 0.49
FFAR1 O14842 1/20 0.48
LMNA P02545 2/20 0.48
TCF4 P15884 1/20 0.48
CTNNB1 P35222 1/20 0.48
MAPK1 P28482 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
POLB P06746 2/20 0.47
HPGD P15428 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
TSHR P16473 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14075324 0.92 KDM4E (0.65) CYP2C9CYP1A2KMT2AMEN1KDM4E
SCHEMBL14075315 0.88 CYP2C9 (0.65) CYP2C9CYP1A2KMT2AMEN1KDM4E
SCHEMBL14075328 0.84 KDM4E (0.61) CYP2C9CYP1A2KMT2AMEN1KDM4E
SCHEMBL14075394 0.84 CYP2C9 (0.78) CYP2C9CYP1A2KMT2AMEN1ALDH1A1
SCHEMBL14075311 0.83 ALDH1A1 (0.74) CYP2C9CYP1A2KMT2AMEN1ALDH1A1
SCHEMBL14075395 0.83 MEN1 (0.65) CYP2C9CYP1A2KMT2AMEN1KDM4E
SCHEMBL14075317 0.81 CYP2C9 (0.69) CYP2C9CYP1A2ALDH1A1CYP2C19POLB
SCHEMBL14075403 0.81 CYP2C9 (0.58) CYP2C9CYP1A2KMT2AMEN1KDM4E
SCHEMBL31504019 0.81 KDM4E (0.72) KMT2AMEN1KDM4EALDH1A1MAPT
SCHEMBL14075346 0.81 CYP2C9 (0.83) CYP2C9CYP1A2KMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7429677-B2 Small molecule entry inhibitors TIBOTEC PHARMACEUTICALS LTD. (IE) 2008-09-30 US disclosed
US-7429677-B2 Small molecule entry inhibitors TIBOTEC PHARMACEUTICALS LTD. (IE) 2008-09-30 US disclosed