SCHEMBL14076366

SCHEMBL14076366

CC(C)(C)c1ccc(OC(C(=O)O)C(=O)O)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.58
SMN1; SMN2 Q16637 2/20 0.53
MAPT P10636 3/20 0.50
TDP1 Q9NUW8 2/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
NR1H4 Q96RI1 1/20 0.47
RAB9A P51151 2/20 0.45
NR4A2 P43354 1/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
RXRA P19793 1/20 0.45
RXRB P28702 1/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
ALOX15 P16050 1/20 0.45
APEX1 P27695 1/20 0.45
MAPK1 P28482 1/20 0.45
RECQL P46063 1/20 0.45
HSD17B10 Q99714 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5272169 0.83 CYP1A2 (0.61) SMN1; SMN2MAPTTDP1L3MBTL1NR1H4
SCHEMBL5273528 0.83 CYP1A2 (0.61) SMN1; SMN2MAPTTDP1L3MBTL1NR1H4
SCHEMBL4343686 0.83 CYP1A2 (0.61) SMN1; SMN2MAPTTDP1L3MBTL1NR1H4
SCHEMBL6693143 0.82 ESR1 (0.53) LDHATDP1RAB9AMEN1KMT2A
SCHEMBL11716060 0.81 SMN1; SMN2 (0.50) SMN1; SMN2MAPTTDP1L3MBTL1NR1H4
SCHEMBL28871353 0.81 SMN1; SMN2 (0.50) SMN1; SMN2MAPTTDP1L3MBTL1NR1H4
SCHEMBL5277876 0.81 SMN1; SMN2 (0.50) SMN1; SMN2MAPTTDP1L3MBTL1NR1H4
SCHEMBL6696803 0.80 LDHA (0.49) LDHASMN1; SMN2MAPTTDP1MEN1
SCHEMBL8935640 0.79 SMN1; SMN2 (0.59) SMN1; SMN2MAPTTDP1L3MBTL1NR1H4
SCHEMBL8935642 0.79 SMN1; SMN2 (0.59) SMN1; SMN2MAPTTDP1L3MBTL1NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080220536-A1 Methods for Identifying Compounds that Modulate Enzymatic Activities by Employing Covalently Bonded Target-Extender Complexes with Ligand Candidates ERIANSON DANIEL A 2008-09-11 US disclosed
US-20080220536-A1 Methods for Identifying Compounds that Modulate Enzymatic Activities by Employing Covalently Bonded Target-Extender Complexes with Ligand Candidates ERIANSON DANIEL A 2008-09-11 US disclosed
US-7214487-B2 Methods for identifying compounds that modulate enzymatic activities by employing covalently bonded target-extender complexes with ligand candidates SUNESIS PHARMACEUTICALS, INC. (US) 2007-05-08 US disclosed
US-7214487-B2 Methods for identifying compounds that modulate enzymatic activities by employing covalently bonded target-extender complexes with ligand candidates SUNESIS PHARMACEUTICALS, INC. (US) 2007-05-08 US disclosed