SCHEMBL14080906

SCHEMBL14080906

NCCOc1ccc(-c2cccnc2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 4/20 0.71
CYP3A4 P08684 3/20 0.71
CYP2D6 P10635 2/20 0.71
CYP2C9 P11712 1/20 0.71
CYP2C19 P33261 1/20 0.71
MKNK1 Q9BUB5 3/20 0.59
MKNK2 Q9HBH9 3/20 0.59
CYP2A6 P11509 3/20 0.57
CYP11B2 P19099 4/20 0.50
CYP11B1 P15538 3/20 0.50
ALDH1A1 P00352 2/20 0.50
CYP1A2 P05177 1/20 0.50
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
MAPT P10636 1/20 0.49
HTT P42858 1/20 0.49
TAAR1 Q96RJ0 1/20 0.48
LTA4H P09960 2/20 0.47
PLA2G2A P14555 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4228524 0.92 CYP19A1 (0.74) CYP19A1CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5751218 0.85 CYP19A1 (0.73) CYP19A1CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL3177161 0.84 MKNK1 (0.56) CYP19A1CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL4861343 0.83 CYP19A1 (0.71) CYP19A1CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL14129887 0.83 CYP2D6 (1.00) CYP19A1CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL12129582 0.82 CYP19A1 (0.69) CYP19A1CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL28046302 0.82 CYP3A4 (0.74) CYP19A1CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL13527207 0.81 CYP2D6 (0.94) CYP19A1CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL31483083 0.80 CHRNB2 (0.62) MKNK2TAAR1LTA4HPLA2G2A
SCHEMBL1622662 0.80 CHRNB2 (0.62) MKNK2TAAR1LTA4HPLA2G2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008106204-A1 MACROLIDE COMPOUNDS AND METHODS OF MAKING AND USING THE SAME RIB-X-PHARMACEUTICALS, INC. (US) 2008-09-04 WO disclosed