SCHEMBL14081848

SCHEMBL14081848

COc1ccc(F)c(/C=C2\SC(=O)NC2=O)c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 3/20 0.68
PIM1 P11309 3/20 0.65
PIM2 Q9P1W9 3/20 0.65
AKR1B1 P15121 2/20 0.65
NPC1 O15118 2/20 0.65
RAB9A P51151 2/20 0.65
IGF1R P08069 1/20 0.59
HPGD P15428 2/20 0.58
LMNA P02545 1/20 0.58
KMT2A Q03164 1/20 0.58
ATM Q13315 1/20 0.57
PTPN1 P18031 2/20 0.54
CA2 P00918 1/20 0.53
POLB P06746 1/20 0.52
CSNK2A2 P19784 1/20 0.52
CLK1 P49759 1/20 0.52
CSNK2B P67870 1/20 0.52
CSNK2A1 P68400 1/20 0.52
DYRK1A Q13627 1/20 0.52
DYRK1B Q9Y463 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7558738 0.87 CA2 (0.71) GSK3BNPC1RAB9AHPGDLMNA
SCHEMBL4801244 0.87 CA2 (0.71) GSK3BNPC1RAB9AHPGDLMNA
SCHEMBL4806036 0.87 CA2 (0.71) GSK3BNPC1RAB9AHPGDLMNA
SCHEMBL15091371 0.85 GSK3B (0.70) GSK3BPIM1PIM2AKR1B1NPC1
SCHEMBL15101838 0.85 GSK3B (0.70) GSK3BPIM1PIM2AKR1B1NPC1
SCHEMBL2541079 0.84 PIM1 (0.69) GSK3BPIM1PIM2AKR1B1NPC1
SCHEMBL2541077 0.84 PIM1 (0.69) GSK3BPIM1PIM2AKR1B1NPC1
SCHEMBL1248964 0.82 CA2 (0.76) GSK3BPIM1PIM2AKR1B1NPC1
SCHEMBL1248963 0.82 CA2 (0.76) GSK3BPIM1PIM2AKR1B1NPC1
SCHEMBL15421728 0.82 CA2 (0.76) GSK3BPIM1PIM2AKR1B1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7417064-B2 3-aryloxy/thio-3-substituted propanamines and their use in inhibiting serotonin and norepinephrine reuptake ELI LILLY AND COMPANY (US) 2008-08-26 US disclosed
US-7417064-B2 3-aryloxy/thio-3-substituted propanamines and their use in inhibiting serotonin and norepinephrine reuptake ELI LILLY AND COMPANY (US) 2008-08-26 US disclosed