SCHEMBL14087635

SCHEMBL14087635

CC1(C)CC(=O)c2cc(N=O)c(NC3CCCC3)nc2C1

nearest known ligand 0.71

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
HTT P42858 1/20 0.50
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4433377 0.83 ALDH1A1 (0.52) ALDH1A1HTTCYP2C19
SCHEMBL14087704 0.83 ALDH1A1 (0.52) ALDH1A1HTTCYP2C19
SCHEMBL4421913 0.80 POLB (0.57) ALDH1A1HTT
SCHEMBL10025783 0.73 ALDH1A1 (0.90) ALDH1A1
SCHEMBL4423510 0.68 ALDH1A1 (0.47) ALDH1A1HTTCYP2C19
SCHEMBL4423861 0.68 POLB (0.51)
SCHEMBL10025798 0.67 ALDH1A1 (1.00) ALDH1A1
SCHEMBL4433327 0.65 POLB (0.53)
SCHEMBL5043832 0.65 ALDH1A1 (0.41) ALDH1A1HTT
SCHEMBL8283793 0.64 ALDH1A1 (0.59) ALDH1A1HTTCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1723116-B1 TETRAHYDROQUINOLINONES AND THEIR USE AS ANTAGONISTS OF METABOTROPIC GLUTAMATE RECEPTORS MERZ PHARMA GMBH & CO KGAA (DE) 2008-09-24 EP disclosed