SCHEMBL14090643

SCHEMBL14090643

CC(=O)Cc1cccc(CC(C)(C)NCC(O)c2ccc(O)c(NS(C)(=O)=O)c2)c1

nearest known ligand 0.77

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 16/20 0.77
ADRB3 P13945 4/20 0.64
CHRM3 P20309 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12305713 1.00 ADRB2 (0.77) ADRB2ADRB3CHRM3
SCHEMBL14620429 0.92 ADRB2 (0.80) ADRB2ADRB3CHRM3
SCHEMBL12305639 0.92 ADRB2 (0.80) ADRB2ADRB3CHRM3
SCHEMBL2450154 0.91 ADRB2 (0.76) ADRB2ADRB3CHRM3
SCHEMBL2450164 0.91 ADRB2 (0.79) ADRB2ADRB3CHRM3
SCHEMBL2450162 0.91 ADRB2 (0.79) ADRB2ADRB3CHRM3
SCHEMBL2450153 0.91 ADRB2 (0.79) ADRB2ADRB3CHRM3
SCHEMBL14204754 0.91 ADRB2 (0.77) ADRB2ADRB3
SCHEMBL12305718 0.89 ADRB2 (0.76) ADRB2ADRB3
SCHEMBL14090671 0.88 ADRB2 (0.61) ADRB2ADRB3CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080193988-A1 Such as 2-(3-{2-[((2R)-2-{4-Benzyloxy-3-[(dimethylsulfonyl)amino]phenyl}-2-{[tert-butyl(dimethyl)silyl]oxy}ethyl)amino]-2-methylpropyl}phenyl)-N-[(4'-hydroxybiphenyl-3-yl)methyl]-acetamide GLADWELL IAIN ROBERT 2008-08-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080193988-A1 Such as 2-(3-{2-[((2R)-2-{4-Benzyloxy-3-[(dimethylsulfonyl)amino]phenyl}-2-{[tert-butyl(dimethyl)silyl]oxy}ethyl)amino]-2-methylpropyl}phenyl)-N-[(4'-hydroxybiphenyl-3-yl)methyl]-acetamide NR4A1, CYP2A6, GPR6 ADRB2 118/4885ADRB3 109/4885CHRM3 257/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.