SCHEMBL14095971

SCHEMBL14095971

COc1cc2ncnc(Nc3ccc(Cl)c(Br)c3)c2cc1OC

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 14/20 0.80
KDR P35968 9/20 0.74
ABCG2 Q9UNQ0 3/20 0.74
JAK3 P52333 2/20 0.74
RET P07949 2/20 0.74
KIF5B P33176 2/20 0.74
ABCB1 P08183 1/20 0.74
FLT1 P17948 1/20 0.71
ERBB2 P04626 4/20 0.71
FBP1 P09467 3/20 0.71
CLK1 P49759 2/20 0.71
EPHB4 P54760 2/20 0.71
AURKA O14965 1/20 0.71
INSR P06213 1/20 0.71
PDGFRB P09619 1/20 0.71
FLT4 P35916 1/20 0.71
TEK Q02763 1/20 0.71
AURKB Q96GD4 1/20 0.71
EPHA2 P29317 2/20 0.70
LCK P06239 4/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14095961 0.90 EGFR (0.80) EGFRKDRABCG2JAK3RET
SCHEMBL5570070 0.89 EGFR (0.85) EGFRKDRABCG2JAK3RET
SCHEMBL2100447 0.89 KDR (0.80) EGFRKDRABCG2RETKIF5B
SCHEMBL5865262 0.86 EGFR (0.81) EGFRKDRABCG2JAK3RET
SCHEMBL22590721 0.86 EGFR (0.80) EGFRKDRABCG2JAK3RET
SCHEMBL6787016 0.85 KDR (0.74) EGFRKDRABCG2JAK3RET
SCHEMBL20812874 0.85 EGFR (0.80) EGFRKDRABCG2JAK3RET
SCHEMBL29711485 0.85 JAK3 (1.00) EGFRKDRABCG2JAK3RET
SCHEMBL29372372 0.85 JAK3 (1.00) EGFRKDRABCG2JAK3RET
SCHEMBL7870579 0.85 KDR (1.00) EGFRKDRABCG2JAK3RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080199480-A1 Methods for Identifying Risk of Type II Diabetes and Treatments Thereof SEQUENOM, INC. (US) 2008-08-21 US disclosed
US-20080199480-A1 Methods for Identifying Risk of Type II Diabetes and Treatments Thereof SEQUENOM, INC. (US) 2008-08-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080199480-A1 Methods for Identifying Risk of Type II Diabetes and Treatments Thereof SLC5A2, GCKR, IAPP EGFR 3981/4885KDR 2859/4885ABCG2 4039/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.