SCHEMBL14098993

SCHEMBL14098993

CC(CO)Cc1c[nH]c2cc(F)c(F)cc12

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 2/20 0.57
HTR2A P28223 6/20 0.49
HTR2C P28335 4/20 0.49
HTR1A P08908 4/20 0.46
HTR2B P41595 4/20 0.46
HTR1D P28221 2/20 0.46
HTR1B P28222 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
NFKB1 P19838 1/20 0.46
CYP2C19 P33261 1/20 0.46
NPSR1 Q6W5P4 2/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
ADRB1 P08588 1/20 0.40
ADRA2A P08913 1/20 0.40
SLC6A2 P23975 1/20 0.40
HTR1E P28566 1/20 0.40
SLC6A4 P31645 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23259357 0.83 GPR84 (0.65) GPR84HTR2AHTR2CHTR1AHTR2B
SCHEMBL30811413 0.82 HTR2A (0.69) GPR84HTR2AHTR2CHTR1AHTR2B
SCHEMBL29280816 0.82 HTR2A (0.69) GPR84HTR2AHTR2CHTR1AHTR2B
SCHEMBL24912883 0.82 HTR2A (0.69) GPR84HTR2AHTR2CHTR1AHTR2B
SCHEMBL5764881 0.82 HTR2A (0.69) GPR84HTR2AHTR2CHTR1ASLC6A4
SCHEMBL13962418 0.82 HTR2A (0.69) GPR84HTR2AHTR2CHTR1ASLC6A4
SCHEMBL4603380 0.81 GPR84 (0.57) GPR84HTR2AHTR2CHTR1AHTR2B
SCHEMBL22122335 0.76 GPR84 (0.59) GPR84HTR2AHTR2CHTR1AHTR2B
SCHEMBL27220736 0.76 GPR84 (0.50) GPR84HTR2AHTR2CHTR1AHTR2B
SCHEMBL27220732 0.76 GPR84 (0.50) GPR84HTR2AHTR2CHTR1AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1956016-A1 Bicyclic acyltryptophanols Bayer Schering Pharma Aktiengesellschaft (DE) 2008-08-13 EP disclosed