SCHEMBL1409980

SCHEMBL1409980

O=CN1C[C@H](NC(=O)c2cc3ccccc3cn2)C(=O)N(CC(=O)N[C@H]2CC(=O)OC2OCc2ccccc2)c2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 17/20 0.46
CASP8 Q14790 11/20 0.38
CASP3 P42574 3/20 0.36
RIPK1 Q13546 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10200557 0.85 CASP1 (0.51) CASP1CASP8CASP3
SCHEMBL13139801 0.85 CASP1 (0.51) CASP1CASP8CASP3
SCHEMBL646831 0.85 CASP1 (0.51) CASP1CASP8CASP3
SCHEMBL645906 0.75 CASP1 (0.65) CASP1CASP8CASP3
SCHEMBL13140322 0.75 CASP1 (0.65) CASP1CASP8CASP3
SCHEMBL645989 0.74 CASP1 (0.69) CASP1CASP8CASP3
SCHEMBL647496 0.74 CASP1 (0.53) CASP1CASP8CASP3
SCHEMBL10201769 0.74 CASP1 (0.68) CASP1CASP8CASP3
SCHEMBL12444062 0.74 CASP1 (0.68) CASP1CASP8CASP3
SCHEMBL10248335 0.73 CASP1 (0.55) CASP1CASP8CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2295442-A2 Inhibitors of interleukin-1beta converting enzyme VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-03-16 EP disclosed