SCHEMBL14105367

SCHEMBL14105367

CN1C(=N)N[C@](C)(c2ccc(F)c(N)c2)[C@H](c2ccc(C(F)(F)F)cc2)C1=O

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
TACR1 P25103 1/20 0.32
BACE1 P56817 1/20 0.31
ESR1 P03372 1/20 0.30
BACE2 Q9Y5Z0 1/20 0.30
AR P10275 1/20 0.30
OPRM1 P35372 1/20 0.30
OPRL1 P41146 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7541540 0.91 MEN1 (0.35) MEN1KMT2ABACE1ESR1AR
SCHEMBL13054967 0.91 MEN1 (0.35) MEN1KMT2ABACE1ESR1AR
SCHEMBL13054594 0.88 ABCC9 (0.35) MEN1KMT2AESR1
SCHEMBL13081820 0.88 MEN1 (0.34) MEN1KMT2AESR1
SCHEMBL7566880 0.88 ABCC9 (0.35) MEN1KMT2AESR1
SCHEMBL7572424 0.85 AR (0.37) MEN1KMT2AAR
SCHEMBL13054170 0.85 AR (0.37) MEN1KMT2AAR
SCHEMBL13054488 0.85 MEN1 (0.37) MEN1KMT2ATACR1ESR1
SCHEMBL7585732 0.85 MEN1 (0.37) MEN1KMT2ATACR1ESR1
SCHEMBL13054304 0.84 BACE1 (0.30) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008103351-A2 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS SCHERING CORPORATION (US) 2008-08-28 WO disclosed