SCHEMBL14110522

SCHEMBL14110522

CN(C)C1(c2ccccc2)CCCCC1c1[nH]c2ccccc2c1CCn1ccnn1

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 7/20 0.37
HTR2C P28335 6/20 0.37
DRD2 P14416 5/20 0.37
OPRM1 P35372 9/20 0.34
OPRL1 P41146 8/20 0.34
SIGMAR1 Q99720 1/20 0.33
OGFRL1 Q5TC84 2/20 0.32
BCHE P06276 1/20 0.32
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL735749 0.83 OPRM1 (0.41) OPRM1OPRL1OGFRL1
SCHEMBL734697 0.77 OPRM1 (0.45) OPRM1OPRL1OGFRL1
SCHEMBL733672 0.73 OPRM1 (0.40) HTR2AHTR2CDRD2OPRM1OPRL1
SCHEMBL734951 0.72 KDM4E (0.43) OPRM1OPRL1OGFRL1KDM4E
SCHEMBL735943 0.70 OPRM1 (0.36) HTR2AHTR2COPRM1OPRL1SIGMAR1
SCHEMBL735790 0.68 OPRM1 (0.41) OPRM1OPRL1OGFRL1
SCHEMBL734685 0.68 OPRM1 (0.41) OPRM1OPRL1OGFRL1
SCHEMBL736060 0.68 OPRM1 (0.48) OPRM1OPRL1OGFRL1
SCHEMBL735200 0.67 HTR2A (0.51) HTR2AHTR2CDRD2OPRM1OPRL1
SCHEMBL734919 0.67 HTR2A (0.52) HTR2AHTR2CDRD2OPRM1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044016-B1 4-HETEROARYL-SUBSTITUTED 1-AMINOCYCLOHEXANE-1-AND CYCLOHEXENE-1-DERIVATIVES HAVING EFFECTS ON THE OPIOD RECEPTOR SYSTEM GRUENENTHAL GMBH (DE) 2012-12-05 EP disclosed