SCHEMBL1411069

SCHEMBL1411069

CC/C(=C\c1ccc(CO)cn1)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.50
L3MBTL1 Q9Y468 3/20 0.50
TBXAS1 P24557 2/20 0.45
CYP3A4 P08684 2/20 0.35
ALDH1A1 P00352 2/20 0.35
NFKB1 P19838 2/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
MAPT P10636 1/20 0.35
PKM P14618 1/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
THPO P40225 1/20 0.35
BLM P54132 1/20 0.35
PMP22 Q01453 1/20 0.35
KMT2A Q03164 1/20 0.35
HIF1A Q16665 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
SMN1; SMN2 Q16637 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1411072 1.00 KDM4E (0.50) KDM4EL3MBTL1TBXAS1CYP3A4ALDH1A1
SCHEMBL1969309 0.80 KDM4E (0.41) KDM4EL3MBTL1TBXAS1MEN1LMNA
SCHEMBL1704854 0.80 TBXAS1 (0.49) KDM4EL3MBTL1TBXAS1CYP3A4ALDH1A1
SCHEMBL1914364 0.80 KDM4E (0.42) KDM4EL3MBTL1TBXAS1ALDH1A1MEN1
SCHEMBL15755442 0.80 TBXAS1 (0.49) KDM4EL3MBTL1TBXAS1CYP3A4ALDH1A1
SCHEMBL16737458 0.80 KDM4E (0.42) KDM4EL3MBTL1TBXAS1ALDH1A1MEN1
SCHEMBL2959588 0.76 TBXAS1 (0.57) TBXAS1CYP3A4CYP2C9PSEN1PSEN2
SCHEMBL11120260 0.73 TDP1 (0.50) KDM4EL3MBTL1TBXAS1ALDH1A1MEN1
SCHEMBL1410986 0.72 EGFR (0.50) KDM4EL3MBTL1TBXAS1CYP3A4ALDH1A1
SCHEMBL1410982 0.72 EGFR (0.50) KDM4EL3MBTL1TBXAS1CYP3A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2295410-A1 HDAC inhibitor Chroma Therapeutics Limited (GB) 2011-03-16 EP disclosed