SCHEMBL14124342

SCHEMBL14124342

N[C@H](CCCNC(=O)OCc1cncs1)Cc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.54
CYP3A4 P08684 18/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14123908 0.88 TDP1 (0.54) TDP1CYP3A4
SCHEMBL18715750 0.87 CYP3A4 (0.65) CYP3A4
SCHEMBL21946533 0.87 CYP3A4 (0.65) CYP3A4
SCHEMBL14123814 0.86 CYP3A4 (0.56) TDP1CYP3A4
SCHEMBL11919313 0.84 RAB9A (0.48) TDP1CYP3A4
SCHEMBL2736231 0.83 CYP3A4 (0.66) CYP3A4
SCHEMBL10067531 0.83 CYP3A4 (0.66) CYP3A4
SCHEMBL18715783 0.83 CYP3A4 (0.66) CYP3A4
SCHEMBL2736188 0.83 CYP3A4 (0.66) CYP3A4
SCHEMBL18715718 0.82 CYP3A4 (0.56) TDP1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008103949-A1 MODULATORS OF PHARMACOKINETIC PROPERTIES OF THERAPEUTICS GILEAD SCIENCES, INC. (US) 2008-08-28 WO disclosed