SCHEMBL14136995

SCHEMBL14136995

C=C(Nc1ccncc1)c1nc(Br)cnc1N

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ATR Q13535 4/20 0.52
PRKCI P41743 3/20 0.47
GRM5 P41594 1/20 0.46
PRKDC P78527 1/20 0.43
TBK1 Q9UHD2 12/20 0.39
IKBKE Q14164 10/20 0.39
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14059993 0.82 ATR (0.76) ATRPRKCIGRM5PRKDCTBK1
SCHEMBL31387927 0.82 ATR (0.76) ATRPRKCIGRM5PRKDCTBK1
SCHEMBL20433220 0.71 MAPKAPK2 (0.52) ATRGRM5PRKDC
SCHEMBL14136996 0.70 ATR (0.50) ATRGRM5PRKDC
SCHEMBL20433296 0.70 ATR (0.71) ATRPRKDCCYP3A4
SCHEMBL559881 0.69 ATR (1.00) ATRGRM5PRKDCCYP3A4
SCHEMBL17418738 0.69 ATR (0.45) ATRGRM5
SCHEMBL15724439 0.69 ATR (0.68) ATRPRKCIGRM5PRKDCCYP3A4
SCHEMBL411951 0.68 ATR (0.75) ATRPRKCIGRM5PRKDCCYP3A4
SCHEMBL1800565 0.67 ATR (0.58) ATRPRKCIGRM5PRKDCCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012161877-A1 PYRIDINE-AND PYRAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2012-11-29 WO disclosed